All targets

Molecular targets of radiopharmaceuticals in clinical trials, with the number of ongoing trials and approved products. Data as of 26 October 2026.

TargetTherapyImagingApproved
PSMA1381085
FAP20101—
Glucose metabolism (FDG)—1121
SSTR 2/371296
Amyloid—331
Neurotransmission (receptors, enzymes)—33—
Amino acid transport—322
Tau—262
CXCR4320—
HER2317—
CAIX710—
TSPO (neuroinflammation)—17—
Bone (bone metastases)15—1
Myocardial perfusion—152
Integrins αvβ3/αvβ658—
Catecholamine synthesis (FDOPA)—131
Cardiac amyloidosis—121
Hypoxia—12—
T-cell activation—11—
Estrogen receptors—111
GRPR64—
CD458——
B7-H362—
Sentinel lymph node—81
Choline (membrane metabolism)—81
PARP—8—
NET (MIBG)7—1
PD-L1 / PD-116—
Synaptic density (SV2A)—7—
Granzyme B—7—
PLE / phospholipid6——
DLL342—
CD8 (T cells)—6—
Proliferation (FLT)—6—
Collagen (fibrosis)—6—
GPC314—
Nectin-414—
Norepinephrine transporter—51
Bone remodelling—5—
Bacteria—5—
α-synuclein—5—
uPAR13—
Cardiac sympathetic innervation—4—
Folate receptor—4—
GLP-1R (exendin)—4—
EGFR—4—
TROP2—4—
Fatty acid metabolism—4—
ACP3 (prostatic acid phosphatase)—4—
Claudin 18.212—
P-glycoprotein (blood–brain barrier)—3—
Thyroid (NIS)—3—
Lung ventilation / perfusion—3—
Dopamine transporter (DAT)—31
Progesterone receptors—3—
Renal function—3—
CD70—3—
CD252——
CEA2——
CD382——
LAT12——
MC1R2——
EGFR / c-MET2——
VAP-1 (vascular inflammation)—2—
Demyelination (K⁺ channels)—2—
EpCAM—2—
Adrenal (CYP11B)—2—
BCMA—2—
Mitochondrial function—2—

A monitoring tool with no regulatory value: check every item at its source.