Radiopharmaceuticals by vector: structure, properties, radiolabelled forms, ongoing trials, approvals and publications. Data as of 27 October 2026.
| Molecule | Target | Radiolabelled forms | Ongoing trials | Approved | Publications |
|---|---|---|---|---|---|
| Fludeoxyglucose | Glucose metabolism (FDG) | ¹⁸F | 113 | ✓ | 60,955 |
| PSMA-617 | PSMA | ¹⁷⁷Lu ²²⁵Ac ¹⁶¹Tb ⁶⁸Ga | 69 | ✓ | 1,264 |
| DOTATATE | SSTR 2/3 | ¹⁷⁷Lu ²²⁵Ac ²¹²Pb ⁶⁸Ga ⁶⁴Cu | 68 | ✓ | 3,170 |
| FAPI-46 | FAP | ⁶⁸Ga ¹⁷⁷Lu | 44 | 341 | |
| PSMA-I&T | PSMA | ¹⁷⁷Lu ²²⁵Ac ¹⁶¹Tb ⁶⁸Ga | 26 | 247 | |
| DCFPyL | PSMA | ¹⁸F | 22 | ✓ | 484 |
| Pentixafor / pentixather | CXCR4 | ⁶⁸Ga ¹⁷⁷Lu ⁹⁰Y | 20 | 384 | |
| PSMA-11 | PSMA | ⁶⁸Ga | 18 | ✓ | 1,345 |
| rhPSMA-7.3 | PSMA | ¹⁸F | 18 | ✓ | 72 |
| DOTATOC | SSTR 2/3 | ¹⁷⁷Lu ⁹⁰Y ⁶⁸Ga | 15 | ✓ | 1,186 |
| Radium dichloride | Bone (bone metastases) | ²²³Ra | 15 | ✓ | 1,380 |
| Fluciclovine | Amino acid transport | ¹⁸F | 14 | ✓ | 486 |
| FDOPA | Catecholamine synthesis (FDOPA) | ¹⁸F | 13 | ✓ | 1,686 |
| Fluoroestradiol | Estrogen receptors | ¹⁸F | 12 | ✓ | 335 |
| Fluoromisonidazole | Hypoxia | ¹⁸F | 12 | 686 | |
| Fluorocholine | Choline (membrane metabolism) | ¹⁸F ¹¹C | 11 | ✓ | 1,535 |
| Flortaucipir | Tau | ¹⁸F | 10 | ✓ | 834 |
| FET | Amino acid transport | ¹⁸F | 9 | ✓ | 691 |
| PSMA-1007 | PSMA | ¹⁸F | 8 | ✓ | 500 |
| FAPI-04 | FAP | ⁶⁸Ga ¹⁸F | 7 | 683 | |
| Iobenguane (MIBG) | Norepinephrine transporter | ¹²³I ¹³¹I | 7 | ✓ | 5,542 |
| FAP-2286 | FAP | ¹⁷⁷Lu ⁶⁸Ga | 6 | 91 | |
| Fluorothymidine | Proliferation (FLT) | ¹⁸F | 6 | 996 | |
| MK-6240 | Tau | ¹⁸F | 5 | ✓ | 145 |
| Sodium fluoride | Bone remodelling | ¹⁸F | 5 | ✓ | 708 |
| NeoB | GRPR | ¹⁷⁷Lu | 3 | 60 | |
| Flutemetamol | Amyloid | ¹⁸F | 3 | ✓ | 440 |
| Florbetapir | Amyloid | ¹⁸F | 1 | ✓ | 1,089 |
| Florbetaben | Amyloid | ¹⁸F | 1 | ✓ | 590 |
| Flurpiridaz | Myocardial perfusion | ¹⁸F | 1 | ✓ | 126 |
| Ioflupane | Neurotransmission (receptors, enzymes) | ¹²³I ¹⁸F | 1 | ✓ | 1,820 |
| Sestamibi | Myocardial perfusion | ⁹⁹ᵐTc | 1 | ✓ | 8,026 |
| Pentetreotide | SSTR 2/3 | ¹¹¹In | — | ✓ | 979 |
| Tetrofosmin | Myocardial perfusion | ⁹⁹ᵐTc | — | ✓ | 1,633 |
| Medronate | Bone remodelling | ⁹⁹ᵐTc | — | ✓ | 1,711 |
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